Publikationen von Herbert Waldmann

Kawamura, T.; Futamura, Y.; Shang, E.; Muroi , M.; Janning, P.; Ueno, M.; Wilke, J.; Takeda, S.; Kondoh , Y.; Ziegler, S. et al.; Watanabe , N.; Waldmann, H.; Osada , H.: Discovery of small-molecule modulator of heterotrimeric G i-protein by integrated phenotypic profiling and chemical proteomics. BioScience, Biotechnology & Biochemistry, S. 1 - 7 (2020)

Grigalunas, M.; Burhop, A.; Christoforow, A.; Waldmann, H.: Pseudo-natural products and natural product-inspired methods in chemical biology and drug discovery. Current Opinion in Chemical Biology 56, S. 111 - 118 (2020)

Shaaban, S.; Davies, C.; Merten, C.; Flegel, J.; Otte, F.; Strohmann, C.; Waldmann, H.: Rh(III)-catalyzed C-H Activation of Aryl-Hydroxamates for the Synthesis of Isoindolinones. Chemistry – A European Journal 26 (47), S. 10729 - 10734 (2020)

Foley, D. J.; Zinken, S.; Corkery, D.; Laraia, L.; Pahl, A.; Wu, Y.-W.; Waldmann, H.: Phenotyping reveals the targets of a pseudo-natural product autophagy inhibitor. Angewandte Chemie, International Edition 59 (11), S. 1 - 17 (2020)

Foley, D. J.; Zinken, S.; Corkery, D.; Laraia, L.; Pahl, A.; Wu, Y.-W.; Waldmann, H.: Phenotyping reveals the targets of a pseudo-natural product autophagy inhibitor. Angewandte Chemie 132 (11), S. 1 - 17 (2020)

Guéret, S. M.; Thavam, S.; Carbajo, R. J.; Potowski, M.; Larsson, N.; Dahl, G.; Dellsén, A.; Grossmann, T. N.; Plowright, A. T.; Valeur, E. et al.; Lemurell, M.; Waldmann, H.: Macrocyclic Modalities Combining Peptide Epitopes and Natural Product Fragments. Journal of the American Chemical Society, S. 1 - 48 (2020)

Karageorgis, G.; Foley, D. J.; Laraia, L.; Waldmann, H.: Principle and design of pseudo-natural products. Nature Chemistry 12 (3), S. 227 - 235 (2020)

Winzker, M.; Friese, A.; Koch, U.; Janning, P.; Ziegler, S.; Waldmann, H.: Development of a PDEδ targeting PROTAC that impairs lipid metabolism. Angewandte Chemie, International Edition 59 (14), S. 5595 - 5601 (2019)

Laraia, L.; Garivet, G.; Foley, D. J.; Kaiser, N.; Müller, S.; Zinken, S.; Pinkert, T.; Wilke, J.; Corkery, D.; Pahl, A. et al.; Sievers, S.; Janning, P.; Arenz, C.; Wu, Y.; Rodriguez, R.; Waldmann, H.: Image-based morphological profiling identifies a lysosomotropic, iron-sequestering autophagy inhibitor. Angewandte Chemie, International Edition 59 (14), S. 5721 - 5729 (2019)

Reckzeh, E. S.; Waldmann, H.: Small Molecule Inhibition of Glucose Transporters GLUT 1‐4. ChemBioChem: A European Journal of Chemical Biology 20, S. 1 - 22 (2019)

Pobbati, A. V.; Mejuch, T.; Chakraborty, S.; Karatas, H.; Bharath, S. R.; Guéret, S. M.; Goy, P.-A.; Hahne, G.; Pahl, A.; Sievers, S. et al.; Guccione, E.; Song, H.; Waldmann, H.; Hong, W.: Identification of Quinolinols as Activators of TEAD-dependent Transcription. ACS Chemical Biology, S. 1 - 35 (2019)

Cromm, P. M.; Adihou, H.; Kapoor, S.; Vazquez-Chantada, M.; Davey, P.; Longmire, D.; Hennes, E.; Hofer, W.; Küchler, P.; Chiarparin, E. et al.; Waldmann, H.; Grossmann, T. N.: Lipidated stapled peptides targeting the acyl binding protein UNC119. ChemBioChem: A European Journal of Chemical Biology, S. 1 - 10 (2019)

Laraia, L.; Garivet, G.; Foley, D. J.; Kaiser, N.; Müller, S.; Zinken, S.; Pinkert, T.; Wilke, J.; Corkery, D.; Pahl, A. et al.; Sievers, S.; Janning, P.; Arenz, C.; Wu, Y.; Rodriguez, R.; Waldmann, H.: Image-based morphological profiling identifies a lysosomotropic, iron-sequestering autophagy inhibitor. Angewandte Chemie 132 (14), S. 5770 - 5778 (2019)

Christoforow, A.; Wilke, J.; Binici, A.; Pahl, A.; Ostermann, C.; Sievers, S.; Waldmann, H.: Design, Synthesis and Phenotypic Profiling of Pyrano-Furo-Pyridone Pseudo Natural Products. Angewandte Chemie International Edition 58 (41), S. 14715 - 14723 (2019)

Reckzeh, E. S.; Karageorgis, G.; Schwalfenberg, M.; Ceballos, J.; Nowacki, J.; Stroet, M. C.M.; Binici, A.; Knauer, L.; Brand, S.; Choidas, A. et al.; Strohmann, C.; Ziegler, S.; Waldmann, H.: Inhibition of Glucose Transporters and Glutaminase Synergistically Impairs Tumor Cell Growth. Cell Chemical Biology 26, S. 1 - 41 (2019)

Ceballos, J.; Schwalfenberg, M.; Karageorgis, G.; Reckzeh, E. S.; Sievers, S.; Ostermann, C.; Pahl, A.; Sellstedt, M.; Nowacki, J.; Carnero Corrales, M. A. et al.; Wilke, J.; Laraia, L.; Tschapalda, K.; Metz, M.; Sehr, D. A.; Brand, S.; Winklhofer, K.; Janning, P.; Ziegler, S.; Waldmann, H.: Synthesis of Indomorphan Pseudo Natural Product Inhibitors of Glucose Transporters GLUT-1 and -3. Angewandte Chemie, International Edition, S. 1 - 28 (2019)

Ceballos, J.; Schwalfenberg, M.; Karageorgis, G.; Reckzeh, E. S.; Sievers, S.; Ostermann, C.; Pahl, A.; Sellstedt, M.; Nowacki, J.; Carnero Corrales, M. A. et al.; Wilke, J.; Laraia, L.; Tschapalda, K.; Metz, M.; Sehr, D. A.; Brand, S.; Winklhofer, K.; Janning, P.; Ziegler, S.; Waldmann, H.: Synthesis of Indomorphan Pseudo Natural Product Inhibitors of Glucose Transporters GLUT‐1 and ‐3. Angewandte Chemie, S. 1 - 28 (2019)

Kremer, L.; Hennes, E.; Brause, A.; Ursu, A.; Robke, L.; Matsubayashi, H. T.; Nihongaki, Y.; Flegel, J.; Mejdrová, I.; Eickhoff, J. et al.; Baumann, M.; Nencka, R.; Janning, P.; Kordes, S.; Schöler, H. R.; Sterneckert, J.; Inoue, T.; Ziegler, S.; Waldmann, H.: Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß. Angewandte Chemie, International Edition, S. 1 - 37 (2019)

Kremer, L.; Hennes, E.; Brause, A.; Ursu, A.; Robke, L.; Matsubayashi , H. T.; Nihongaki, Y.; Flegel, J.; Mejdrová, I.; Eickhoff, J. et al.; Baumann, M.; Nencka, R.; Janning, P.; Kordes, S.; Schöler, H. R.; Sterneckert, J.; Inoue, T.; Ziegler, S.; Waldmann, H.: Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß. Angewandte Chemie, S. 1 - 37 (2019)

Furuta, T.; Mizukami, Y.; Asano, L.; Kotake, K.; Ziegler, S.; Yoshida, H.; Watanabe, M.; Sato, S.-i.; Waldmann, H.; Nishikawa, M. et al.; Uesugi, M.: Nutrient-Based Chemical Library as a Source of Energy Metabolism Modulators. ACS Chemical Biology, S. 1 - 6 (2019)