Publikationen von Daniel Rauh

Zeitschriftenartikel (50)

Zeitschriftenartikel
Becker, C.; Öcal, S.; Nguyen, H. D.; Phan, T.; Keul, M.; Simard, J. R.; Rauh, D.: Monitoring Conformational Changes in the Receptor Tyrosine Kinase EGFR. ChemBioChem: A European Journal of Chemical Biology 17 (11), S. 990 - 994 (2016)
Zeitschriftenartikel
Fang, Z.; Simard, J. R.; Plenker, D.; Nguyen, H. D.; Phan, T.; Wolle, P.; Baumeister, S.; Rauh, D.: Discovery of Inter-Domain Stabilizers-A Novel Assay System for Allosteric Akt Inhibitors. ACS Chemical Biology 10 (1), S. 279 - 288 (2015)
Zeitschriftenartikel
Richters, A.; Nguyen, H. D.; Phan, T.; Simard, J. R.; Grütter, C.; Engel, J.; Rauh, D.: Identification of Type II and III DDR2 Inhibitors. Journal of Medicinal Chemistry 57 (10), S. 4252 - 4262 (2014)
Zeitschriftenartikel
Richters, A.; Ketzer, J.; Getlik, M.; Grütter, C.; Schneider, R.; Heuckmann, J. M.; Heynck, S.; Sos, M. L.; Gupta, A.; Unger, A. et al.; Schultz-Fademrecht, C.; Thomas, R. K.; Bauer, S.; Rauh, D.: Targeting Gain of Function and Resistance Mutations in Abl and KIT by Hybrid Compound Design. Journal of Medicinal Chemistry 56 (14), 1, S. 5757 - 5772 (2013)
Zeitschriftenartikel
Schneider, R.; Gohla, A.; Simard, J. R.; Yadav, D. B.; Fang, Z.; van Otterlo, W. A. L.; Rauh, D.: Overcoming Compound Fluorescence in the FLiK Screening Assay with Red-Shifted Fluorophores. Journal of the American Chemical Society 135 (22), 1, S. 8400 - 8408 (2013)
Zeitschriftenartikel
Schneider, R.; Beumer, C.; Simard, J. R.; Grütter, C.; Rauh, D.: Selective Detection of Allosteric Phosphatase Inhibitors. Journal of the American Chemical Society 135 (18), 1, S. 6838 - 6841 (2013)
Zeitschriftenartikel
Over, B.; Wetzel, S.; Grütter, C.; Nakai, Y.; Renner, S.; Rauh, D.; Waldmann, H.: Natural-product-derived fragments for fragment-based ligand discovery. Nature Chemistry 5 (1), 1, S. 21 - 28 (2013)
Zeitschriftenartikel
Sos, M. L.; Dietlein, F.; Peifer, M.; Schöttle, J.; Balke-Want, H.; Müller, C.; Koker, M.; Richters, A.; Heynck, S.; Malchers, F. et al.; Heuckmann, J. M.; Seidel, D.; Eyers, P. A.; Ullrich, R. T.; Antonchick, A. P.; Vintonyak, V. V.; Schneider, P. M.; Ninomiya, T.; Waldmann, H.; Büttner, R.; Rauh, D.; Heukamp, L. C.; Thomas, R. K.: A framework for identification of actionable cancer genome dependencies in small cell lung cancer. Proceedings of the National Academy of Sciences of the United States of America 109 (42), 1, S. 17034 - 17039 (2012)
Zeitschriftenartikel
Getlik, M.; Simard, J. R.; Termathe, M.; Grütter, C.; Rabiller, M.; Van Otterlo, W. A. L.; Rauh, D.: Fluorophore Labeled Kinase Detects Ligands That Bind within the MAPK Insert of p38α Kinase. PLoS ONE 7 (7), 1, S. e39713-1 - e39713-10 (2012)
Zeitschriftenartikel
Schneider, R.; Becker, C.; Simard, J. R.; Getlik, M.; Bohlke, N.; Janning, P.; Rauh, D.: Direct Binding Assay for the Detection of Type IV Allosteric Inhibitors of Abl. Journal of the American Chemical Society 134 (22), 1, S. 9138 - 9141 (2012)
Zeitschriftenartikel
Grütter, C.; Simard, J. R.; Mayer-Wrangowski, S. C.; Schreier, P. H.; Pérez-Martín, J.; Richters, A.; Getlik, M.; Gutbrod, O.; Braun, C. A.; Beck, M. E. et al.; Rauh, D.: Targeting GSK3 from Ustilago maydis: Type-II Kinase Inhibitors as Potential Antifungals. ACS Chemical Biology 7 (7), 1, S. 1257 - 1267 (2012)
Zeitschriftenartikel
Koch, A.; Rode, H. B.; Richters, A.; Rauh, D.; Hauf, S.: A Chemical Genetic Approach for Covalent Inhibition of Analogue-Sensitive Aurora Kinase. ACS Chemical Biology 7 (4), 1, S. 723 - 731 (2012)
Zeitschriftenartikel
Antonchick, A. P.; Schuster, H.; Bruss, H.; Schürmann, M.; Preut, H.; Rauh, D.; Waldmann, H.: Enantioselective synthesis of the spirotryprostatin A scaffold. Tetrahedron 67 (52), 1, S. 10195 - 10202 (2011)
Zeitschriftenartikel
Vintonyak, V. V.; Warburg, K.; Over, B.; Hübel, K.; Rauh, D.; Waldmann, H.: Identification and further development of thiazolidinones spiro-fused to indolin-2-ones as potent and selective inhibitors of Mycobacterium tuberculosis protein tyrosine phosphatase B. Tetrahedron 67 (35), 1, S. 6713 - 6729 (2011)
Zeitschriftenartikel
Tückmantel, S.; Greul, J. N.; Janning, P.; Brockmeyer, A.; Grütter, C.; Simard, J. R.; Gutbrod, O.; Beck, M. E.; Tietjen, K.; Rauh, D. et al.; Schreier, P. H.: Identification of Ustilago maydis Aurora Kinase As a Novel Antifungal Target. Asc Chemical Biology 6 (9), 1, S. 926 - 933 (2011)
Zeitschriftenartikel
Rode, H. B.; Sos, M. L.; Grütter, C.; Heynck, S.; Simard, J. R.; Rauh, D.: Synthesis and biological evaluation of 7-substituted-1-(3-bromophenylamino)isoquinoline-4-carbonitriles as inhibitors of myosin light chain kinase and epidermal growth factor receptor. Bioorganic & Medicinal Chemistry 19 (1), 1, S. 429 - 439 (2011)
Zeitschriftenartikel
Vintonyak, V. V.; Waldmann, H.; Rauh, D.: Using small molecules to target protein phosphatases. Bioorganic & Medicinal Chemistry 19 (7), 1, S. 2145 - 2155 (2011)
Zeitschriftenartikel
Klüter, S.; Simard, J. R.; Rode, H. B.; Grütter, C.; Pawar, V.; Raaijmakers, H. C. A.; Barf, T. A.; Rabiller, M.; van Otterlo, W. A. L.; Rauh, D.: Characterization of Irreversible Kinase Inhibitors by Directly Detecting Covalent Bond Formation: A Tool for Dissecting Kinase Drug Resistance. ChemBioChem 11 (18), 1, S. 2557 - 2566 (2010)
Zeitschriftenartikel
Robubi, A.; Waldmann, H.; Rauh, D.: RAF Kinase Inhibitors in Cancer Treatment: Like a Bull in a China Shop? ChemBioChem 11 (12), 1, S. 1645 - 1648 (2010)
Zeitschriftenartikel
Vintonyak, V. V.; Warburg, K.; Kruse, H.; Grimme, S.; Hübel, K.; Rauh, D.; Waldmann, H.: Identification of Thiazolidinones Spiro-Fused to Indolin-2-ones as Potent and Selective Inhibitors of the Mycobacterium tuberculosis Protein Tyrosine Phosphatase B. Angewandte Chemie 122 (34), 1, S. 6038 - 6041 (2010)
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