Publications of Herbert Waldmann

Lumbierres, M.; Palomo, J. M.; Kragol, G.; Roehrs, S.; Müller, O.; Waldmann, H.: Solid-Phase Synthesis of Lipidated Peptides. Chemistry - A European Journal 11 (24), 1, pp. 7405 - 7415 (2005)

Vogel, A.; Katzka, C. P.; Waldmann, H.; Arnold, K.; Brown, M. F.; Huster, D.: Lipid Modifications of a Ras Peptide Exhibit Altered Packing and Mobility versus Host Membrane as Detected by ²H Solid-State NMR. Journal of the American Chemical Society 127 (35), 1, pp. 12263 - 12272 (2005)

Deck, P.; Pendzialek, D.; Biel, M.; Wagner, M.; Popkirova, B.; Ludolph, B.; Kragol, G.; Kuhlmann, J.; Athanassios, G.; Waldmann, H.: Development and Biological Evaluation of Acyl Protein Thioesterase 1 (APT1) Inhibitors. Angewandte Chemie International Edition 44 (31), 1, pp. 4975 - 4980 (2005)

Deck, P.; Pendzialek, D.; Biel, M.; Wagner, M.; Popkirova, B.; Ludolph, B.; Kragol, G.; Kuhlmann, J.; Athanassios, G.; Waldmann, H.: Development and Biological Evaluation of Acyl Protein Thioesterase 1 (APT1) Inhibitors. Angewandte Chemie 117 (31), 1, pp. 5055 - 5060 (2005)

Dekker, F. J.; Koch, M. A.; Waldmann, H.: Protein structure similarity clustering (PSSC) and natural product structure as inspiration sources for drug development and chemical genomics. Current Opinion in Chemical Biology 9 (3), 1, pp. 232 - 239 (2005)

Bialy, L.; Waldmann, H.: Inhibitoren der Proteintyrosinphosphatasen: Kandidaten für zukünftige Wirkstoffe? Angewandte Chemie 117 (25), 1, pp. 3880 - 3906 (2005)

Bialy, L.; Waldmann, H.: Inhibitors of Protein Tyrosine Phosphatases: Next-Generation Drugs? Angewandte Chemie International Edition 44 (25), 1, pp. 3814 - 3839 (2005)

Manger, M.; Scheck, M.; Prinz, H.; von Kries, J. P.; Langer, T.; Saxena, K.; Schwalbe, H.; Fürstner, A.; Rademann, J.; Waldmann, H.: Discovery of Mycobacterium Tuberculosis Protein Tyrosine Phosphatase A (MptpA) Inhibitors Based on Natural Products and a Fragment-Based Approach. ChemBioChem 6 (10), 1, pp. 1749 - 1753 (2005)

Balamurugan, R.; Dekker, F. J.; Waldmann, H.: Design of compound libraries based on natural product scaffolds and protein structure similarity clustering (PSSC). Molecular BioSystems 1 (1), 1, pp. 36 - 45 (2005)

Koch, M. A.; Waldmann, H.: Protein structure similarity clustering and natural product structure as guiding principles in drug discovery. Drug Discovery Today 10 (7), 1, pp. 471 - 483 (2005)

Rocks, O.; Peyker, A.; Kahms, M.; Verveer, P. J.; Koerner, C.; Lumbierres, M.; Kuhlmann, J.; Waldmann, H.; Wittinghofer, A.; Bastiaens, P. I. H.: An Acylation Cycle Regulates Localization and Activity of Palmitoylated Ras Isoforms. Science 307 (5716), 1, pp. 1746 - 1752 (2005)

Brunsveld, L.; Watzke, A.; Durek, T.; Alexandrov, K.; Goody, R. S.; Waldmann, H.: Synthesis of Functionalized Rab GTPases by a Combination of Solution- or Solid-Phase Lipopeptide Synthesis with Expressed Protein Ligation. Chemistry - A European Journal 11 (9), 1, pp. 2756 - 2772 (2005)

Watzke, A.; Brunsveld, L.; Durek, T.; Alexandrov, K.; Rak, A.; Goody, R. S.; Waldmann, H.: Chemical biology of protein lipidation: semi-synthesis and structure elucidation of prenylated RabGTPases. Organic & Biomolecular Chemistry 3 (7), 1, pp. 1157 - 1164 (2005)

Gourzoulidou, E.; Carpintero, M.; Baumhof, P.; Giannis, A.; Waldmann, H.: Inhibition of Angiogenesis-Relevant Receptor Tyrosine Kinases by Sulindac Analogues. ChemBioChem 6 (3), 1, pp. 527 - 531 (2005)

Rosenbaum, C.; Röhrs, S.; Müller, O.; Waldmann, H.: Modulation of MRP-1-Mediated Multidrug Resistance by Indomethacin Analogues. Journal of Medicinal Chemistry 48 (4), 1, pp. 1179 - 1187 (2005)

Reents, R.; Wagner, M.; Schlummer, S.; Kuhlmann, J.; Waldmann, H.: Synthesis and Application of Fluorescent Ras Proteins for Live-Cell Imaging. ChemBioChem 6 (1), 1, pp. 86 - 94 (2005)

Bayer, E.; Thutewohl, M.; Christner, C.; Tradler, T.; Osterkamp, F.; Waldmann, H.; Bayer, P.: Idenfication of hPin1 inhibitors that induce apoptosis in a mammalian Ras transformed cell line. Chemical Communications 2005, 1, pp. 516 - 518 (2005)

Dursina, B.-E.; Reents, R.; Niculae, A.; Veligodsky, A.; Breitling, R.; Pyatkov, K.; Waldmann, H.; Goody, R. S.; Alexandrov, K.: A genetically encodable microtag for chemo-enzymatic derivatization and purification of recombinant proteins. Protein Expression and Purification 39 (1), 1, pp. 71 - 81 (2005)

Goody, R. S.; Durek, T.; Waldmann, H.; Brunsveld, L.; Alexandrov, K.: Application of Protein Semisynthesis for the Construction of Functionalized Posttranslationally modified Rab GTPases. GTPases Regulating Membrane Targeting and Fusion, 4, pp. 29 - 42 (2005)

Sommer, S.; Waldmann, H.: Solid phase synthesis of a spiro[5.5]ketal library. Chemical Communications 45, 1, pp. 5684 - 5686 (2005)