Publications of Herbert Waldmann

Müller, O.; Gourzoulidou, E.; Carpintero, M.; Karaguni, I.-M.; Langerak, A.; Herrmann, C.; Möröy, T.; Klein-Hitpass, L.; Waldmann, H.: Identification of potent Ras signaling inhibitors by pathway-selective phenotype-based screening. Angewandte Chemie 116 (4), 1, pp. 456 - 460 (2004)

Rosenbaum, C.; Baumhof, P.; Mazitscheck, R.; Müller, O.; Giannis, A.; Waldmann, H.: Synthesis and Biological Evaluation of an Indomethacin Library Reveals a New Class of Angiogenesis-Related Kinase Inhibitors. Angewandte Chemie 116 (2), 1, pp. 226 - 230 (2004)

Rosenbaum, C.; Baumhof, P.; Mazitschek, R.; Müller, O.; Giannis, A.; Waldmann, H.: Synthesis and biological evaluation of an indomethacin library reveals a new class of angiogenesis-related kinase inhibitors. Angewandte Chemie-International Edition 43 (2), 1, pp. 224 - 228 (2004)

Waldmann, H.; Karaguni, I.-M.; Carpintero, M.; Gourzoulidou, E.; Herrmann, C.; Brockmann, C.; Oschkinat, H.; Müller, O.: Sulindac-derived Ras pathway inhibitors target the Ras-Raf interaction and downstream effectors in the Ras pathway. Angewandte Chemie-International Edition 43 (4), 1, pp. 454 - 458 (2004)

Waldmann, H.; Karaguni, I.-M.; Carpintero, M.; Gourzoulidou, E.; Herrmann, C.; Brockmann, C.; Oschkinat, H.; Müller, O.: Sulindac-derived Ras pathway inhibitors target the Ras-Raf interaction and downstream effectors in the Ras pathway. Angewandte Chemie 116 (4), 1, pp. 460 - 464 (2004)

Fürstner, A.; Feyen, F.; Prinz, H.; Waldmann, H.: Total Synthesis and Reassessment of the Phosphatase- Inhibitory Activity of the Antitumor Agent TMC-69-6H. Angewandte Chemie 115 (43), 1, pp. 5519 - 5522 (2003)

Gerdes, J. M.; Waldmann, H.: Direct mass spectrometric monitoring of solid phase organic syntheses. Journal of Combinatorial Chemistry 5 (6), 1, pp. 814 - 820 (2003)

Waldmann, H.: At the crossroads of chemistry and biology. Bioorganic & Medicinal Chemistry 11 (14), 1, pp. 3045 - 3051 (2003)

Bialy, L.; Waldmann, H.: Synthesis and biological evaluation of cytostatin analogues. Chemical Communications 2003 (15), 1, pp. 1872 - 1873 (2003)

Fürstner, A.; Feyen, F.; Prinz, H.; Waldmann, H.: Total synthesis and reassessment of the phosphatase-inhibitory activity of the antitumor agent TMC-69-6H. Angewandte Chemie-International Edition 42 (43), 1, pp. 5361 - 5364 (2003)

Huster, D.; Vogel, A.; Katzka, C.; Scheidt, H. A.; Binder, H.; Dante, S.; Gutberlet, T.; Zschörnig, O.; Waldmann, H.; Arnold, K.: Membrane insertion of a lipidated ras peptide studied by FTIR, solid-state NMR, and neutron diffraction spectroscopy. Journal of the American Chemical Society 125 (14), 1, pp. 4070 - 4079 (2003)

Kissau, L.; Stahl, P.; Mazitschek, R.; Giannis, A.; Waldmann, H.: Development of natural product-derived receptor tyrosine kinase inhibitors based on conservation of protein domain fold. Journal of Medicinal Chemistry 46 (14), 1, pp. 2917 - 2931 (2003)

Koch, M. A.; Breinbauer, R.; Waldmann, H.: Protein structure similarity as guiding principle for combinatorial library design. Biological Chemistry 384 (9), 1, pp. 1265 - 1272 (2003)

Köhn, M.; Wacker, R.; Peters, C.; Schröder, H.; Soulère, L.; Breinbauer, R.; Niemeyer, C. M.; Waldmann, H.: Staudinger ligation: A new immobilization strategy for the preparation of small-molecule arrays. Angewandte Chemie-International Edition 42 (47), 1, pp. 5830 - 5834 (2003)

Köhn, M.; Wacker, R.; Peters, C.; Schröder, H.; Soulère, L.; Breinbauer, R.; Niemeyer, C. M.; Waldmann, H.: Staudinger-Ligation: eine Immobilisierungsstrategie zur Herstellung von Wirkstoff-Arrays. Angewandte Chemie 115 (47), 1, pp. 6010 - 6014 (2003)

Ludolph, B.; Waldmann, H.: The synthesis of acid- and base-labile lipopeptides on solid support. Chemistry-A European Journal 9 (15), 1, pp. 3683 - 3691 (2003)

Peters, C.; Waldmann, H.: Solid-phase synthesis of peptide esters employing the hydrazide linker. Journal of Organic Chemistry 68 (15), 1, pp. 6053 - 6055 (2003)

Pylypenko, O.; Rak, A.; Reents, R.; Niculae, A.; Sidorovitch, V.; Cioaca, M.-D.; Bessolitsyna, E.; Thomä, N. H.; Waldmann, H.; Schlichting, I. et al.; Goody, R. S.; Alexandrov, K.: Structure of rab escort protein-1 in complex with Rab geranylgeranyltransferase. Molecular Cell 11 (2), 1, pp. 483 - 494 (2003)

Rak, A.; Pylypenko, O.; Durek, T.; Watzke, A.; Kushnir, S.; Brunsveld, L.; Waldmann, H.; Goody, R. S.; Alexandrov, K.: Structure of Rab GDP-dissociation inhibitor in complex with prenylated YPT1 GTPase. Science 302 (5645), 1, pp. 646 - 650 (2003)

Rosenbaum, C.; Katzka, C.; Marzinzik, A.; Waldmann, H.: Traceless Fischer indole synthesis on the solid phase. Chemical Communications 2003 (15), 1, pp. 1822 - 1823 (2003)