Publications of Herbert Waldmann

Stieber, F.; Grether, U.; Mazitschek, R.; Soric, N.; Giannis, A.; Waldmann, H.: Multistep solid-phase synthesis of an antibiotic and receptor tyrosine kinase inhibitors using the traceless phenylhydrazide linker. Chemistry-A European Journal 9 (14), 1, pp. 3282 - 3291 (2003)

Stieber, F.; Grether, U.; Waldmann, H.: Development of the traceless phenylhydrazide linker for solid-phase synthesis. Chemistry-A European Journal 9 (14), 1, pp. 3270 - 3281 (2003)

Thutewohl, M.; Kissau, L.; Popkirova, B.; Karaguni, I.-M.; Nowak, T.; Bate, M.; Kuhlmann, J.; Müller, O.; Waldmann, H.: Identification of mono- and bisubstrate inhibitors of protein farnesyltransferase and inducers of apoptosis from a pepticinnamin E library. Bioorganic & Medicinal Chemistry 11 (12), 1, pp. 2617 - 2626 (2003)

Thutewohl, M.; Waldmann, H.: Solid-phase synthesis of a pepticinnamin E library. Bioorganic & Medicinal Chemistry 11 (12), 1, pp. 2591 - 2615 (2003)

Völkert, M.; Uwai, K.; Tebbe, A.; Popkirova, B.; Wagner, M.; Kuhlmann, J.; Waldmann, H.: Synthesis and biological activity of photoactivatable N-Ras peptides and proteins. Journal of the American Chemical Society 125 (42), 1, pp. 12749 - 12758 (2003)

Waldmann, H.: Natürlich kombinatorisch - naturstoffgetriebene Wirkstoffentwicklung. Nachrichten aus der Chemie 51 (2), 1, pp. 126 - 131 (2003)

Waldmann, H.; Breinbauer, R.; Koch, M. A.: Naturstoffgetriebene kombinatorische Chemie. Postgenomics - vom Molekül zur Funktion, 1, pp. 478 - 479 (2003)

Stieber, F.; Mazitschek, R.; Soric, N.; Giannis, A.; Waldmann, H.: Traceless solid-phase synthesis of 2-aminothiazoles: Receptor tyrosine kinase inhibitors with dual selectivity for tie-2 and VEGFR-2. Angewandte Chemie - International Edition 41 (24), 1, pp. 4757 - 4761 (2002)

Stieber, F.; Mazitschek, R.; Soric, N.; Giannis, A.; Waldmann, H.: Festphasensynthese von 2-Aminothiazolen unter Verwendung des spurlosen Hydrazid-Ankers: Rezeptortyrosinkinase-Inhibitoren mit dualer Selektivität für Tie-2 und VEGFR-2. Angewandte Chemie 114 (24), 1, pp. 4951 - 4955 (2002)

Breinbauer, R.; Manger, M.; Scheck, M.; Waldmann, H.: Natural product guided compound library development. Current Medicinal Chemistry 9 (23), 1, pp. 2129 - 2145 (2002)

Brohm, D.; Philippe, N.; Metzger, S.; Bhargava, A.; Müller, O.; Lieb, F.; Waldmann, H.: Solid-phase synthesis of dysidiolide-derived protein phosphatase inhibitors. Journal of the American Chemical Society 124 (44), 1, pp. 13171 - 13178 (2002)

Waldmann, H.; Breinbauer, R.: Nature provides the answer. Natural product structures as guiding principle in combinatorial chemistry. Screening: Trends in Drug Discovery 3 (6), 1, pp. 46 - 48 (2002)

Huttenloch, O.; Laxman, E.; Waldmann, H.: Solid-Phase Development of Chiral Phosphoramidite Ligands for Enantioselective Conjugate Addition Reactions. Chemistry - A European Journal 8 (20), 1, pp. 4767 - 4780 (2002)

Thutewohl, M.; Kissau, L.; Popkirova, B.; Karaguni, I.-M.; Nowak, T.; Bate, M.; Kuhlmann, J.; Müller, O.; Waldmann, H.: Festphasensynthese und biologische Evaluierung einer Pepticinnamin-E-Bibliothek. Angewandte Chemie 114 (19), 1, pp. 3768 - 3772 (2002)

Völkert, M.; Koul, S.; Müller, G. H.; Lehnig, M.; Waldmann, H.: Phenylhydrazide as an enzyme-labile protecting group in peptide synthesis. Journal of Organic Chemistry 67 (20), 1, pp. 6902 - 6910 (2002)

Peters, C.; Wagner, M.; Völkert, M.; Waldmann, H.: Bridging the gap between cell biology and organic chemistry: chemical synthesis and biological application of lipidated peptides and proteins. Naturwissenschaften 89 (9), 1, pp. 381 - 390 (2002)

Ludolph, B.; Eisele, F.; Waldmann, H.: Solution- and solid-phase synthesis of the polybasic lipid-modified C termini of Rho A and K-Ras 4B. ChemBioChem 3 (9), 1, pp. 901 - 904 (2002)

Breinbauer, R.-P.; Vetter, I. R.; Waldmann, H.: Von Proteindomänen zu Wirkstoffkandidaten - Naturstoffe als Leitstrukturen für das Design und die Synthese von Substanzbibliotheken. Angewandte Chemie 114 (16), 1, pp. 3002 - 3015 (2002)

Eisele, F.; Kuhlmann, J.; Waldmann, H.: Synthesis and membrane binding properties of a lipopeptide fragment from influenza virus A hemagglutinin. Chemistry - A European Journal 8 (15), 1, pp. 3362 - 3376 (2002)

Ludolph, B.; Eisele, F.; Waldmann, H.: Solid-Phase Synthesis of Lipidated Peptides. Journal of the American Chemical Society 124 (21), 1, pp. 5954 - 5955 (2002)