Publikationen von Herbert Waldmann

Ludolph, B.; Waldmann, H.: Solid-phase synthesis of benzodiazepinediones mimicking the C-terminus of the H-Ras protein. Tetrahedron Letters 50 (26), 1, S. 3148 - 3150 (2009)

Oprea, T. I.; Bologa, C. G.; Boyer, S.; Curpan, R. F.; Glen, R. C.; Hopkins, A. L.; Lipinski, C. A.; Marshall, G. R.; Martin, Y. C.; Ostopovici-Halip, L. et al.; Rishton, G.; Ursu, O.; Vaz, R. J.; Waller, C.; Waldmann, H.; Sklar, L. A.: A crowdsourcing evaluation of the NIH chemical probes. Nature Chemical Biology 5 (7), 1, S. 441 - 447 (2009)

Renner, S.; Van Otterlo, W. A. L.; Dominguez Seoane, M.; Möcklinghoff, S.; Hofmann, B.; Wetzel, S.; Schuffenhauer, A.; Ertl, P.; Oprea, T. I.; Steinhilber, D. et al.; Brunsveld, L.; Rauh, D.; Waldmann, H.: Bioactivity-guided mapping and navigation of chemical space. Nature Chemical Biology 5 (8), 1, S. 585 - 592 (2009)

Wetzel, S.; Klein, K.; Renner, S.; Rauh, D.; Oprea, T. I.; Mutzel, P.; Waldmann, H.: Interactive Exploration of Chemical Space with Scaffold Hunter. Nature Chemical Biology 5 (8), 1, S. 581 - 583; 696 (2009)

Vintonyak, V. V.; Antonchick, A. P.; Rauh, D.; Waldmann, H.: The therapeutic potential of phosphatase inhibitors. Current Opinion in Chemical Biology 13 (3), 1, S. 272 - 283 (2009)

Siegel, G.; Obernosterer, G.; Fiore, R.; Oehmen, M.; Bicker, S.; Christensen, M.; Khudayberdiev, S.; Leuschner, P. F.; Busch, C. J. L.; Kane, C. et al.; Hübel, K.; Dekker, F.; Hedberg, C.; Rengarajan, B.; Drepper, C.; Waldmann, H.; Kauppinen, S.; Greenberg, M. E.; Draguhn, A.; Rehmsmeier, M.; Martinez, J.; Schratt, G. M.: A functional screen implicates microRNA-138-dependent regulation of the depalmitoylation enzyme APT1 in dendritic spine morphogenesis. Nature Cell Biology 11 (6), 1, S. 705 - 716 (2009)

Walther, T.; Renner, S.; Waldmann, H.; Arndt, H.-D.: Synthesis and Structure-Activity Correlation of a Brunsvicamide-Inspired Cyclopeptide Collection. ChemBioChem 10 (7), 1, S. 1153 - 1162 (2009)

Nguyen, U. T. T.; Guo, Z.; Delon, C.; Wu, Y.; Deraeve, C.; Fränzel, B.; Bon, R. S.; Blankenfeldt, W.; Goody, R. S.; Waldmann, H. et al.; Wolters, D.; Alexandrov, K.: Analysis of the eukaryotic prenylome by isoprenoid affinity tagging. Nature Chemical Biology 5 (4), 1, S. 227 - 237 (2009)

Yoshida, M.; Hedberg, C.; Kaiser, M.; Waldmann, H.: Traceless solid phase synthesis of natural product inspired cis-1,2-dehydrodecalins. Chemical Communications 2009 (20), 1, S. 2926 - 2928 (2009)

Kumar, K.; Waldmann, H.: Synthesis of Natural Product Inspired Compound Collections. Angewandte Chemie International Edition 48 (18), 1, S. 3224 - 3242 (2009)

Kumar, K.; Waldmann, H.: Die Synthese von naturstoffinspirierten Verbindungsbibliotheken. Angewandte Chemie 121 (18), 1, S. 3272 - 3290 (2009)

Bulic, B.; Pickhardt, M.; Schmidt, B.; Mandelkow, E. M.; Waldmann, H.; Mandelkow, E.: Entwicklung von Inhibitoren der Tau-Aggregation bei Morbus Alzheimer. Angewandte Chemie 121 (10), 1, S. 1772 - 1785 (2009)

Bulic, B.; Pickhardt, M.; Schmidt, B.; Mandelkow, E.-M.; Waldmann, H.; Mandelkow, E.: Development of Tau Aggregation Inhibitors for Alzheimer's Disease. Angewandte Chemie International Edition 48 (10), 1, S. 1740 - 1752 (2009)

Triola, G.; Wetzel, S.; Ellinger, B.; Koch, M. A.; Hübel, K.; Rauh, D.; Waldmann, H.: ATP competitive inhibitors of D-alanine-D-alanine ligase based on protein kinase inhibitor scaffolds. Bioorganic & Medicinal Chemistry 17 (3), 1, S. 1079 - 1087 (2009)

Waldmann, H.: Killing 84 birds with one stone. Nature Chemical Biology 5 (2), 1, S. 76 - 77 (2009)

Alexander, M.; Gerauer, M.; Pechlivanis, M.; Popkirova, B.; Dvorsky, R.; Brunsveld, L.; Waldmann, H.; Kuhlmann, J.: Mapping the Isoprenoid Binding Pocket of PDEδ by a Semisynthetic, Photoactivatable N-Ras Lipoprotein. ChemBioChem 10 (1), 1, S. 98 - 108 (2009)

Brunsveld, L.; Waldmann, H.; Huster, D.: Membrane binding of lipidated Ras peptides and proteins - The structural point of view. Biochimica et Biophysica Acta - Biomembranes 1788 (1), 1, S. 273 - 288 (2009)

Tan, K.-T.; Guiu-Rozas, E.; Bon, R. S.; Guo, Z.; Delon, C.; Wetzel, S.; Arndt, S.; Alexandrov, K.; Waldmann, H.; Goody, R. S. et al.; Wu, Y.-W.; Blankenfeldt, W.: Design, Synthesis, and Characterization of Peptide-Based Rab Geranylgeranyl Transferase Inhibitors. Journal of Medicinal Chemistry 52 (24), 1, S. 8025 - 8037 (2009)

Tannert, R.; Hu, T.-S.; Arndt, H.-D.; Waldmann, H.: Solid-phase based total synthesis of Jasplakinolide by ring-closing metathesis. Chemical Communications 2009 (12), 1, S. 1493 - 1495 (2009)

Weise, K.; Triola, G.; Brunsveld, L.; Waldmann, H.; Winter, R.: Influence of the Lipidation Motif on the Partitioning and Association of N-Ras in Model Membrane Subdomains. Journal of the American Chemical Society 131 (4), 1, S. 1557 - 1564 (2009)