Publications of Eyad K. Fansa
All genres
Journal Article (18)
1.
Journal Article
26 (6), pp. 842 - 851 (2019)
Small-Molecule Inhibition of the UNC-Src Interaction Impairs Dynamic Src Localization in Cells. Cell Chemical Biology 2.
Journal Article
399 (3), pp. 277 - 292 (2017)
Mechanism and dynamics of INPP5E transport into and inside the ciliary compartment. Biological Chemistry 3.
Journal Article
24 (5), pp. 589 - 597 (2017)
Covalent Protein Labeling at Glutamic Acids. Cell chemical biology 4.
Journal Article
56, pp. 1 - 7 (2017)
Small-Molecule Inhibition of the UNC119–Cargo Interaction. Angewandte Chemie International Edition 5.
Journal Article
129, pp. 1 - 7 (2017)
Small-Molecule Inhibition of the UNC119–Cargo Interaction. Angewandte Chemie 6.
Journal Article
56 (9), pp. 2423 - 2428 (2017)
A PDE6δ-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2. Angewandte Chemie International Edition 7.
Journal Article
129 (9), pp. 2463 - 2468 (2017)
A PDE6d-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2. Angewandte Chemie 8.
Journal Article
398 (5-6), pp. 535 - 545 (2016)
Structure-based development of PDEδ inhibitors. Biological Chemistry 9.
Journal Article
291 (51), pp. 26364 - 26376 (2016)
IQGAP1 Interaction with RHO Family Proteins Revisited KINETIC AND EQUILIBRIUM EVIDENCE FOR MULTIPLE DISTINCT BINDING SITES. The Journal of Biological Chemistry 10.
Journal Article
291 (39), pp. 20766 - 20778 (2016)
Novel biochemical and structural insights into the interaction of myristoylated cargo with Unc119 and their release by Arl2/3. The Journal of Biological Chemistry 11.
Journal Article
7, 11360, pp. 1 - 9 (2016)
Identification of pyrazolopyridazinones as PDEδ inhibitors. Nature Communications 12.
Journal Article
6, 24165, pp. 1 - 16 (2016)
Galectin-1 dimers can scaffold Raf-effectors to increase H-ras nanoclustering. Scientific Reports 13.
Journal Article
7, 11366, pp. 1 - 9 (2016)
PDE6δ-mediated sorting of INPP5E into the cilium is determined by cargo-carrier affinity. Nature Communications 14.
Journal Article
7 (4), pp. 222 - 230 (2016)
Sorting of lipidated cargo by the Arl2/Arl3 system. Small GTPases 15.
Journal Article
23 (25), pp. 6083 - 6093 (2016)
Development of Pyridazinone Chemotypes Targeting the PDEδ Prenyl Binding Site. Chemistry – A European Journal 16.
Journal Article
16 (12), pp. 1583 - 1585 (2015)
The N- and C-terminal ends of RPGR can bind to PDE6δ. EMBO Reports 17.
Journal Article
109 (8), pp. 1619 - 1629 (2015)
Effect of the N-Terminal Helix and Nucleotide Loading on the Membrane and Effector Binding of Arl2/3. Biophysical Journal 18.
Journal Article
15 (13), pp. 1991 - 1997 (2014)
Predicted incorporation of non-native substrates by a polyketide synthase yields bioactive natural product derivatives. ChemBioChem: A European Journal of Chemical Biology