Publications of Herbert Waldmann

Laraia, L.; Waldmann, H.: Natural product inspired compound collections: evolutionary principle, chemical synthesis, phenotypic screening, and target identification. Drug Discovery Today: Technologies 23, pp. 75 - 82 (2017)

Jia, Z.-J.; Merten , C.; Gontla, R.; Daniliuc, C. G.; Antonchick, A. P.; Waldmann, H.: General Enantioselective C−H Activation with Efficiently Tunable Cyclopentadienyl Ligands. Angewandte Chemie 129 (9), pp. 2469 - 2474 (2017)

Jia, Z.-J.; Merten, C.; Gontla, R.; Daniliuc, C. G.; Antonchick, A. P.; Waldmann, H.: General Enantioselective C-H Activation with Efficiently Tunable Cyclopentadienyl Ligands. Angewandte Chemie International Edition 56 (9), pp. 2429 - 2434 (2017)

Lee, Y.-C.; Patil, S.; Golz, C.; Strohmann, C.; Ziegler, S.; Kumar, K.; Waldmann, H.: A ligand-directed divergent catalytic approach to establish structural and functional scaffold diversity. Nature Communications 8, 14043 (2017), pp. 1 - 12 (2017)

Martín-Gago, P.; Fansa, E. K.; Klein, C.; Murarka, S.; Janning, P.; Schürmann, M.; Metz, M.; Ismail, S.; Schultz-Fademrecht, C.; Baumann, M. et al.; Bastiaens, P. I. H.; Wittinghofer, A.; Waldmann, H.: A PDE6δ-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2. Angewandte Chemie International Edition 56 (9), pp. 2423 - 2428 (2017)

Martín-Gago, P.; Fansa, E. K.; Klein, C.; Murarka, S.; Janning, P.; Schürmann, M.; Metz, M.; Ismail, S.; Schultz-Fademrecht, C.; Baumann, M. et al.; Bastiaens, P. I. H.; Wittinghofer, A.; Waldmann, H.: A PDE6d-KRas Inhibitor Chemotype with up to Seven H-Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2. Angewandte Chemie 129 (9), pp. 2463 - 2468 (2017)

Laraia, L.; Ohsawa, K.; Konstantinidis, G.; Robke, L.; Wu, Y.-W.; Kumar, K.; Waldmann, H.: Discovery of Novel Cinchona-Alkaloid-Inspired Oxazatwistane Autophagy Inhibitors. Angewandte Chemie International Edition 56 (8), pp. 2145 - 2150 (2017)

Laraia, L.; Ohsawa, K.; Konstantinidis, G.; Robke, L.; Wu, Y.-W.; Kumar, K.; Waldmann, H.: Discovery of Novel Cinchona-Alkaloid-Inspired Oxazatwistane Autophagy Inhibitors. Angewandte Chemie 129 (8), pp. 2177 - 2182 (2017)

Lee, Y.-C.; Kumar, K.; Waldmann, H.: Ligandengesteuerte divergente Synthese von carbo‐ und heterocyclischen Ringsystemen. Angewandte Chemie 130 (19), pp. 5308 - 5322 (2017)

Murarka, S.; Golz, C.; Strohmann, C.; Antonchick, A. P.; Waldmann, H.: Biology-Oriented Synthesis of 3,3-Spiro(2-tetrahydrofuranyl)oxindoles. Synthesis 49 (1), pp. 87 - 95 (2017)

Martín-Gago, P.; Fansa, E. K.; Wittinghofer, A.; Waldmann, H.: Structure-based development of PDEδ inhibitors. Biological Chemistry 398 (5-6), pp. 535 - 545 (2016)

Schröder, P.; Bauer, J. O.; Strohmann, C.; Kumar, K.; Waldmann, H.: Synthesis of an Iridoid-Inspired Compound Collection and Discovery of Autophagy Inhibitors. The Journal of Organic Chemistry 81 (21), pp. 10242 - 10255 (2016)

Jaiswal, M.; Fansa, E. K.; Kösling, S. K.; Mejuch, T.; Waldmann, H.; Wittinghofer, A.: Novel biochemical and structural insights into the interaction of myristoylated cargo with Unc119 and their release by Arl2/3. The Journal of Biological Chemistry 291 (39), pp. 20766 - 20778 (2016)

Cromm, P. M.; Spiegel, J.; Küchler, P.; Dietrich, L.; Kriegesmann, J.; Wendt, M.; Goody, R. S.; Waldmann, H.; Grossmann, T.: Protease-resistant and cell-permeable double-stapled peptides targeting the Rab8a GTPase. ACS Chemical Biology 11 (8), pp. 2375 - 2382 (2016)

Mejuch, T.; Waldmann, H.: Synthesis of Lipidated Proteins. Bioconjugate Chemistry 27 (8), pp. 1771 - 1783 (2016)

Sperlich, B.; Kapoor, S.; Waldmann, H.; Winter, R.; Weise, K.: Regulation of K-Ras4B Membrane Binding by Calmodulin. Biophysical Journal 111 (1), pp. 113 - 122 (2016)

Perez Galan, P.; Waldmann, H.; Kumar, K.: Building polycyclic indole scaffolds via gold(I)-catalyzed intra- and inter-molecular cyclization reactions of 1,6-enynes. Tetrahedron 72 (26), pp. 3647 - 3652 (2016)

Kötzner, L.; Leutzsch, M.; Sievers, S.; Patil, S.; Waldmann, H.; Zheng, Y.; Thiel, W.; List, B.: The Organocatalytic Approach to Enantiopure 2H- and 3H-Pyrroles: Inhibitors of the Hedgehog Signaling Pathway. Angewandte Chemie International Edition 55 (27), pp. 7693 - 7697 (2016)

Kötzner, L.; Leutzsch, M.; Sievers, S.; Patil, S.; Waldmann, H.; Zheng, Y.; Thiel, W.; List, B.: Organokatalytische Synthese von enantiomerenreinen 2H- und 3H-Pyrrolen: Inhibitoren des Hedgehog-Signalwegs. Angewandte Chemie 128 (27), pp. 7824 - 7828 (2016)

Qian, Y.; Schürmann, M.; Janning, P.; Hedberg, C.; Waldmann, H.: Activity-Based Proteome Profiling Probes Based on Woodward's Reagent K with Distinct Target Selectivity. Angewandte Chemie 128 (27), pp. 7897 - 7902 (2016)