Publications of Daniel Rauh
All genres
Journal Article (50)
Journal Article
2 (9), 1, pp. 735 - 740 (2010)
Highly enantioselective synthesis and cellular evaluation of spirooxindoles inspired by natural products. Nature Chemistry
Journal Article
132 (12), 1, pp. 4152 - 4160 (2010)
Fluorophore Labeling of the Glycine-Rich Loop as a Method of Identifying Inhibitors That Bind to Active and Inactive Kinase Conformations. Journal of the American Chemical Society
Journal Article
6 (6), 1, pp. 449 - 456 (2010)
Small-molecule inhibition of APT1 affects Ras localization and signaling. Nature Chemical Biology
Journal Article
53 (7), 1, pp. 2892 - 2901 (2010)
Synthesis and Biological Evaluation of 4-Anilinoquinolines as Potent Inibitors of Epidermal Growth Factor Receptor. Journal of Medicinal Chemistry
Journal Article
58 (2), 1, pp. 118 - 121 (2010)
Inaktive Kinasekonformationen stabilisieren. Nachrichten aus der Chemie
Journal Article
5 (1), 1, p. e8919 (2010)
Analysis of Compound Synergy in High-Throughput Cellular Screens by Population-Based Lifetime Modeling. PLoS ONE
Journal Article
53 (1), 1, pp. 357 - 367 (2010)
Displacement Assay for the Detection of Stabilizers of Inactive Kinase Conformations. Journal of Medicinal Chemistry
Journal Article
343 (4), 1, pp. 193 - 206 (2010)
Proteus in the World of Proteins: Conformational Changes in Protein Kinases. Archiv der Pharmazie
Journal Article
58 (2), 1, pp. 118 - 122 (2010)
Inaktive Kinasekonformationen stabilisieren. Nachrichten aus der Chemie
Journal Article
70 (3), 1, pp. 868 - 874 (2010)
Chemogenomic Profiling Provides Insights into the Limited Activity of Irreversible EGFR Inhibitors in Tumor Cells Expressing the T790M EGFR Resistance Mutation. Cancer Research
Journal Article
49 (34), 1, pp. 5902 - 5905 (2010)
Identification of Thiazolidinones Spiro-Fused to Indolin-2-ones as Potent and Selective Inhibitors of the Mycobacterium tuberculosis Protein Tyrosine Phosphatase B. Angewandte Chemie International Edition
Journal Article
49 (21), 1, pp. 3666 - 3670 (2010)
A Scaffold-Tree-Merging Strategy for Prospective Bioactivity Annotation of γ-Pyrones. Angewandte Chemie International Edition
Journal Article
106 (43), 1, pp. 18351 - 18356 (2009)
Identifying genotype-dependent efficacy of single and combined PI3K- and MAPK-pathway inhibition in cancer. Proceedings of the National Academy of Sciences of the United States of America
Journal Article
4 (11), 1, pp. 1793 - 1795 (2009)
Chemical and Structural Biology to Direct the Repurposing of Sulindac. ChemMedChem
Journal Article
131 (37), 1, pp. 13286 - 13296 (2009)
Development of a Fluorescent-Tagged Kinase Assay System for the Detection and Characterization of Allosteric Kinase Inhibitors. Journal of the American Chemical Society
Journal Article
5 (8), 1, pp. 585 - 592 (2009)
Bioactivity-guided mapping and navigation of chemical space. Nature Chemical Biology
Journal Article
5 (8), 1, pp. 581 - 583; 696 (2009)
Interactive Exploration of Chemical Space with Scaffold Hunter. Nature Chemical Biology
Journal Article
13 (3), 1, pp. 272 - 283 (2009)
The therapeutic potential of phosphatase inhibitors. Current Opinion in Chemical Biology
Journal Article
52 (13), 1, pp. 3915 - 3926 (2009)
Hybrid Compound Design to Overcome the Gatekeeper T338M Mutation in cSrc. Journal of Medicinal Chemistry
Journal Article
5 (6), 1, pp. 394 - 396 (2009)
A new screening assay for allosteric inhibitors of cSrc. Nature Chemical Biology