Publications of Herbert Waldmann

Foley, D. J.; Zinken, S.; Corkery, D.; Laraia, L.; Pahl, A.; Wu, Y.-W.; Waldmann, H.: Phenotyping reveals the targets of a pseudo-natural product autophagy inhibitor. Angewandte Chemie, International Edition 59 (11), pp. 1 - 17 (2020)

Foley, D. J.; Zinken, S.; Corkery, D.; Laraia, L.; Pahl, A.; Wu, Y.-W.; Waldmann, H.: Phenotyping reveals the targets of a pseudo-natural product autophagy inhibitor. Angewandte Chemie 132 (11), pp. 1 - 17 (2020)

Guéret, S. M.; Thavam, S.; Carbajo, R. J.; Potowski, M.; Larsson, N.; Dahl, G.; Dellsén, A.; Grossmann, T. N.; Plowright, A. T.; Valeur, E. et al.; Lemurell, M.; Waldmann, H.: Macrocyclic Modalities Combining Peptide Epitopes and Natural Product Fragments. Journal of the American Chemical Society, pp. 1 - 48 (2020)

Karageorgis, G.; Foley, D. J.; Laraia, L.; Waldmann, H.: Principle and design of pseudo-natural products. Nature Chemistry 12 (3), pp. 227 - 235 (2020)

Winzker, M.; Friese, A.; Koch, U.; Janning, P.; Ziegler, S.; Waldmann, H.: Development of a PDEδ targeting PROTAC that impairs lipid metabolism. Angewandte Chemie, International Edition 59 (14), pp. 5595 - 5601 (2019)

Laraia, L.; Garivet, G.; Foley, D. J.; Kaiser, N.; Müller, S.; Zinken, S.; Pinkert, T.; Wilke, J.; Corkery, D.; Pahl, A. et al.; Sievers, S.; Janning, P.; Arenz, C.; Wu, Y.; Rodriguez, R.; Waldmann, H.: Image-based morphological profiling identifies a lysosomotropic, iron-sequestering autophagy inhibitor. Angewandte Chemie, International Edition 59 (14), pp. 5721 - 5729 (2019)

Reckzeh, E. S.; Waldmann, H.: Small Molecule Inhibition of Glucose Transporters GLUT 1‐4. ChemBioChem: A European Journal of Chemical Biology 20, pp. 1 - 22 (2019)

Pobbati, A. V.; Mejuch, T.; Chakraborty, S.; Karatas, H.; Bharath, S. R.; Guéret, S. M.; Goy, P.-A.; Hahne, G.; Pahl, A.; Sievers, S. et al.; Guccione, E.; Song, H.; Waldmann, H.; Hong, W.: Identification of Quinolinols as Activators of TEAD-dependent Transcription. ACS Chemical Biology, pp. 1 - 35 (2019)

Cromm, P. M.; Adihou, H.; Kapoor, S.; Vazquez-Chantada, M.; Davey, P.; Longmire, D.; Hennes, E.; Hofer, W.; Küchler, P.; Chiarparin, E. et al.; Waldmann, H.; Grossmann, T. N.: Lipidated stapled peptides targeting the acyl binding protein UNC119. ChemBioChem: A European Journal of Chemical Biology, pp. 1 - 10 (2019)

Laraia, L.; Garivet, G.; Foley, D. J.; Kaiser, N.; Müller, S.; Zinken, S.; Pinkert, T.; Wilke, J.; Corkery, D.; Pahl, A. et al.; Sievers, S.; Janning, P.; Arenz, C.; Wu, Y.; Rodriguez, R.; Waldmann, H.: Image-based morphological profiling identifies a lysosomotropic, iron-sequestering autophagy inhibitor. Angewandte Chemie 132 (14), pp. 5770 - 5778 (2019)

Christoforow, A.; Wilke, J.; Binici, A.; Pahl, A.; Ostermann, C.; Sievers, S.; Waldmann, H.: Design, Synthesis and Phenotypic Profiling of Pyrano-Furo-Pyridone Pseudo Natural Products. Angewandte Chemie International Edition 58 (41), pp. 14715 - 14723 (2019)

Reckzeh, E. S.; Karageorgis, G.; Schwalfenberg, M.; Ceballos, J.; Nowacki, J.; Stroet, M. C.M.; Binici, A.; Knauer, L.; Brand, S.; Choidas, A. et al.; Strohmann, C.; Ziegler, S.; Waldmann, H.: Inhibition of Glucose Transporters and Glutaminase Synergistically Impairs Tumor Cell Growth. Cell Chemical Biology 26, pp. 1 - 41 (2019)

Ceballos, J.; Schwalfenberg, M.; Karageorgis, G.; Reckzeh, E. S.; Sievers, S.; Ostermann, C.; Pahl, A.; Sellstedt, M.; Nowacki, J.; Carnero Corrales, M. A. et al.; Wilke, J.; Laraia, L.; Tschapalda, K.; Metz, M.; Sehr, D. A.; Brand, S.; Winklhofer, K.; Janning, P.; Ziegler, S.; Waldmann, H.: Synthesis of Indomorphan Pseudo Natural Product Inhibitors of Glucose Transporters GLUT-1 and -3. Angewandte Chemie, International Edition, pp. 1 - 28 (2019)

Ceballos, J.; Schwalfenberg, M.; Karageorgis, G.; Reckzeh, E. S.; Sievers, S.; Ostermann, C.; Pahl, A.; Sellstedt, M.; Nowacki, J.; Carnero Corrales, M. A. et al.; Wilke, J.; Laraia, L.; Tschapalda, K.; Metz, M.; Sehr, D. A.; Brand, S.; Winklhofer, K.; Janning, P.; Ziegler, S.; Waldmann, H.: Synthesis of Indomorphan Pseudo Natural Product Inhibitors of Glucose Transporters GLUT‐1 and ‐3. Angewandte Chemie, pp. 1 - 28 (2019)

Kremer, L.; Hennes, E.; Brause, A.; Ursu, A.; Robke, L.; Matsubayashi, H. T.; Nihongaki, Y.; Flegel, J.; Mejdrová, I.; Eickhoff, J. et al.; Baumann, M.; Nencka, R.; Janning, P.; Kordes, S.; Schöler, H. R.; Sterneckert, J.; Inoue, T.; Ziegler, S.; Waldmann, H.: Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß. Angewandte Chemie, International Edition, pp. 1 - 37 (2019)

Kremer, L.; Hennes, E.; Brause, A.; Ursu, A.; Robke, L.; Matsubayashi , H. T.; Nihongaki, Y.; Flegel, J.; Mejdrová, I.; Eickhoff, J. et al.; Baumann, M.; Nencka, R.; Janning, P.; Kordes, S.; Schöler, H. R.; Sterneckert, J.; Inoue, T.; Ziegler, S.; Waldmann, H.: Discovery of the Hedgehog Pathway Inhibitor Pipinib that Targets PI4KIIIß. Angewandte Chemie, pp. 1 - 37 (2019)

Furuta, T.; Mizukami, Y.; Asano, L.; Kotake, K.; Ziegler, S.; Yoshida, H.; Watanabe, M.; Sato, S.-i.; Waldmann, H.; Nishikawa, M. et al.; Uesugi, M.: Nutrient-Based Chemical Library as a Source of Energy Metabolism Modulators. ACS Chemical Biology, pp. 1 - 6 (2019)

Laraia, L.; Friese, A.; Corkery, D. P.; Konstantinidis, G.; Erwin, N.; Hofer, W.; Karatas, H.; Klewer, L.; Brockmeyer, A.; Metz, M. et al.; Schölermann, B.; Dwivedi, M.; Li, L.; Rios-Munoz, P.; Köhn, M.; Winter, R.; Vetter, I. R.; Ziegler, S.; Janning, P.; Wu, Y.-W.; Waldmann, H.: The cholesterol transfer protein GRAMD1A regulates autophagosome biogenesis. Nature Chemical Biology 15 (7), pp. 710 - 720 (2019)

Garivet, G.; Hofer, W.; Konitsiotis, A.; Klein, C.; Kaiser, N.; Mejuch, T.; Fansa, E. K.; Alsaabi, R.; Wittinghofer, A.; Bastiaens, P. I. H. et al.; Waldmann, H.: Small-Molecule Inhibition of the UNC-Src Interaction Impairs Dynamic Src Localization in Cells. Cell Chemical Biology 26 (6), pp. 842 - 851 (2019)

Friese, A.; Ursu, A.; Hochheimer, A.; Schöler, H. R.; Waldmann, H.; Bruder, J. M.: The Convergence of Stem Cell Technologies and Phenotypic Drug Discovery. Cell Chemical Biology 26 (8), pp. 1050 - 1066 (2019)