Publications of Herbert Waldmann

Kaiser, N.; Corkery, D.; Wu, Y.; Laraia, L.; Waldmann, H.: Modulation of autophagy by the novel mitochondrial complex I inhibitor Authipyrin. Bioorganic & Medicinal Chemistry 27 (12 (SI)), pp. 2444 - 2448 (2019)

Friese, A.; Kapoor, S.; Schneidewind, T.; Rao Vidadala, S.; Sardana, J.; Brause, A.; Förster, T.; Bischoff, M.; Wagner, J.; Janning, P. et al.; Ziegler, S.; Waldmann, H.: Chemical genetics reveals a role of dCTP pyrophosphatase 1 in Wnt signaling. Angewandte Chemie International Edition, pp. 1 - 14 (2019)

Friese, A.; Kapoor, S.; Schneidewind, T.; Rao Vidadala, S.; Sardana, J.; Brause, A.; Förster, T.; Bischoff, M.; Wagner, J.; Janning, P. et al.; Ziegler, S.; Waldmann, H.: Chemical genetics reveals a role of dCTP pyrophosphatase 1 in Wnt signaling. Angewandte Chemie, pp. 1 - 14 (2019)

Förster, T.; Shang, E.; Shimizu, K.; Sanada, E.; Schölermann, B.; Hübecker, M.; Hahne, G.; Pascual Lopez-Alberca, M.; Janning, P.; Watanabe, N. et al.; Sievers, S.; Giordanetto, F.; Shimizu, T.; Ziegler, S.; Osada, H.; Waldmann, H.: 2-Sulfonylpyrimidines Target the Kinesin HSET via Cysteine Alkylation. European Journal of Organic Chemistry, pp. 1 - 12 (2019)

Schneidewind, T.; Kapoor, S.; Garivet, G.; Karageorgis, G.; Narayan, R.; Vendrell Navarro, G.; Antonchick, A. P.; Ziegler, S.; Waldmann, H.: The Pseudo Natural Product Myokinasib Is a Myosin Light Chain Kinase 1 Inhibitor with Unprecedented Chemotype. Cell Chemical Biology 26 (4), pp. 512 - 523 (2019)

Nemec, V.; Hylsová, M.; Maier, L.; Flegel, J.; Sievers, S.; Ziegler, S.; Schröder, M.; Berger, B.-T.; Chaikuad, A.; Valcíková, B. et al.; Uldrijan, S.; Drápela, S.; Soucek, K.; Waldmann, H.; Knapp, S.; Paruch, K.: Furo[3,2-b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway. Angewandte Chemie International Edition 58 (4), pp. 1062 - 1066 (2019)

Nemec, V.; Hylsová, M.; Maier, L.; Flegel, J.; Sievers, S.; Ziegler, S.; Schröder, M.; Berger, B.-T.; Chaikuad, A.; Valcíková, B. et al.; Uldrijan, S.; Drápela, S.; Soucek, K.; Waldmann, H.; Knapp, S.; Paruch, K.: Furo[3,2-b]pyridine: A Privileged Scaffold for Highly Selective Kinase Inhibitors and Effective Modulators of the Hedgehog Pathway. Angewandte Chemie 131 (4), pp. 1074 - 1078 (2019)

`T Hart, P.; Openy, J.; Krzyzanowski, A.; Adihou, H.; Waldmann, H.: Hot-spot guided design of macrocyclic inhibitors of the LSD1-CoREST1 interaction. Tetrahedron 75 (48), 130685, pp. 1 - 11 (2019)

Christoforow, A.; Wilke, J.; Binici, A.; Pahl, A.; Ostermann, C.; Sievers, S.; Waldmann, H.: Design, Synthesis and Phenotypic Profiling of Pyrano-Furo-Pyridone Pseudo Natural Products. Angewandte Chemie 131 (41), pp. 14857 - 14865 (2019)

Karageorgis, G.; Waldmann, H.: Guided by Evolution: Biology-Oriented Synthesis of Bioactive Compound Classes. Synthesis 51 (1), pp. 55 - 66 (2019)

Kumar, K.; Waldmann, H.: Nature Inspired Small Molecules for Chemical Biology. Israel Journal of Chemistry 59 (1-2), pp. 41 - 51 (2019)

Reckzeh, E. S.; Waldmann, H.: Development of Glucose Transporter (GLUT) Inhibitors. European Journal of Organic Chemistry, pp. 1 - 10 (2019)

Winzker, M.; Friese, A.; Koch, U.; Janning, P.; Ziegler, S.; Waldmann, H.: Development of a PDEd targeting PROTAC that impairs lipid metabolism. Angewandte Chemie 132 (14), pp. 5644 - 5650 (2019)

Wu, Y.-W.; Waldmann, H.: Toward the role of cholesterol and cholesterol transfer protein in autophagosome biogenesis. Autophagy 15 (12), pp. 2167 - 2168 (2019)

Li, H.; Gontla, R.; Flegel, J.; Merten , C.; Ziegler, S.; Antonchick, A. P.; Waldmann, H.: Enantioselective Formal C(sp3 )-H Bond Activation in the Synthesis of Bioactive Spiropyrazolone Derivatives. Angewandte Chemie International Edition 58 (1), pp. 307 - 311 (2018)

Karageorgis, G.; Reckzeh, E. S.; Ceballos, J.; Schwalfenberg, M.; Sievers, S.; Ostermann, C.; Pahl, A.; Ziegler, S.; Waldmann, H.: Chromopynones are pseudo natural product glucose uptake inhibitors targeting glucose transporters GLUT-1 and -3. Nature Chemistry 10, pp. 1103 - 1111 (2018)

Lee, Y.-C.; Knauer, L.; Louven, K.; Golz, C.; Strohmann, C.; Waldmann, H.; Kumar, K.: Gold(I)-Catalyzed and Nucleophile-Guided Ligand-Directed Divergent Synthesis. European Journal of Organic Chemistry (41), pp. 5688 - 5699 (2018)

Jia, Z.-J.; Shan, G.; Daniliuc, C. G.; Antonchick, A. P.; Waldmann, H.: Enantioselective Synthesis of the Spiro-Tropanyl Oxindole Scaffold Through Bimetallic Relay Catalysis. Angewandte Chemie International Edition 57 (44), pp. 14493 - 14497 (2018)

Jia, Z.-J.; Shan, G.; Daniliuc, C. G.; Antonchick, A. P.; Waldmann, H.: Enantioselective Synthesis of the Spiro-Tropanyl Oxindole Scaffold Through Bimetallic Relay Catalysis. Angewandte Chemie 130 (44), pp. 14701 - 14705 (2018)

Shan, G.; Flegel, J.; Li, H.; Merten, C.; Ziegler, S.; Antonchick, A. P.; Waldmann, H.: C-H Bond Activation for the Synthesis of Heterocyclic Atropisomers Yields Hedgehog Pathway Inhibitors. Angewandte Chemie International Edition 57 (43), pp. 14250 - 14254 (2018)