Publications of Herbert Waldmann

Hennes, E.; Lampe, P.; Dötsch, L.; Bruning, N.; Pulvermacher, L.-M.; Sievers, S.; Ziegler, S.; Waldmann, H.: Cell‐Based Identification of New IDO1 Modulator Chemotypes. Angewandte Chemie International Edition 60 (18), pp. 9869 - 9874 (2021)

Hennes, E.; Lampe, P.; Dötsch, L.; Bruning, N.; Pulvermacher, L.-M.; Sievers, S.; Ziegler, S.; Waldmann, H.: Cell-Based Identification of New IDO1 Modulator Chemotypes. Angewandte Chemie 133 (18), pp. 9957 - 9962 (2021)

Grigalunas, M.; Burhop, A.; Zinken, S.; Pahl, A.; Gally, J.-M.; Wild, N.; Mantel, Y.; Sievers, S.; Foley, D. J.; Scheel, R. et al.; Strohmann, C.; Antonchick, A. P.; Waldmann, H.: Natural product fragment combination to performance-diverse pseudo-natural products. Nature Communications 12 (1), 1883, pp. 1 - 11 (2021)

Ziegler, S.; Sievers, S.; Waldmann, H.: Morphological profiling of small molecules. Cell Chemical Biology 28 (3), pp. 300 - 319 (2021)

Krzyzanowski, A.; Gasper, R.; Adihou, H.; `T Hart, P.; Waldmann, H.: Biochemical Investigation of the Interaction of pICln, RioK1 and COPR5 with the PRMT5-MEP50 Complex. Chembiochem 22 (11), pp. 1908 - 1914 (2021)

Wilke, J.; Kawamura, T.; Xu, H.; Brause, A.; Friese, A.; Metz, M.; Schepmann, D.; Wünsch, B.; Artacho-Cordón, A.; Nieto, F. R. et al.; Watanabe, N.; Osada, H.; Ziegler, S.; Waldmann, H.: Discovery of a σ 1 receptor antagonist by combination of unbiased cell painting and thermal proteome profiling. Cell Chemical Biology 28, pp. 1 - 13 (2021)

Shaaban, S.; Li, H.; Merten, C.; Antonchick, A. P.; Waldmann, H.: Rhodium(III)-Catalyzed Enantioselective Benzamidation of Cyclopropenes. Synthesis 53, pp. 1 - 9 (2021)

Shaaban, S.; Li, H.; Otte, F.; Strohmann, C.; Antonchick, A. P.; Waldmann, H.: Enantioselective Synthesis of Five-Membered-Ring Atropisomers with a Chiral Rh(III) Complex. Organic Letters 22 (23), pp. 9199 - 9202 (2020)

Cremosnik, G. S.; Liu, J.; Waldmann, H.: Guided by evolution: from biology oriented synthesis to pseudo natural products. Natural Product Reports 37 (11), pp. 1497 - 1510 (2020)

Liu, J.; Cremosnik, G. S.; Otte, F.; Pahl, A.; Sievers, S.; Strohmann, C.; Waldmann, H.: Design, synthesis and biological evaluation of chemically and biologically diverse pyrroquinoline pseudo natural products. Angewandte Chemie International Edition 60 (9), pp. 4648 - 4656 (2020)

Schneidewind, T.; Brause, A.; Pahl, A.; Burhop, A.; Mejuch, T.; Sievers, S.; Waldmann, H.; Ziegler, S.: Morphological profiling enables the identification of common mode of action for small molecules with different targets. Chembiochem 21 (22), pp. 3197 - 3207 (2020)

Liu, J.; Cremosnik, G. S.; Otte, F.; Pahl, A.; Sievers, S.; Strohmann, C.; Waldmann, H.: Design, synthesis and biological evaluation of chemically and biologically diverse pyrroquinoline pseudo natural products. Angewandte Chemie 133 (9), pp. 4698 - 4706 (2020)

Adihou, H.; Gopalakrishnan, R.; Förster, T.; Guéret, S. M.; Gasper, R.; Geschwindner, S.; Carrillo García , C.; Karatas, H.; Pobbati, A. V.; Vazquez-Chantada, M. et al.; Davey, P.; Wassvik, C. M.; Pang, J. K. S.; Soh, B. S.; Hong, W.; Chiarparin, E.; Schade, D.; Plowright, A. T.; Valeur, E.; Lemurell, M.; Grossmann, T. N.; Waldmann, H.: A protein tertiary structure mimetic modulator of the Hippo signalling pathway. Nature Communications 11 (1), 5425, pp. 1 - 10 (2020)

Karatas, H.; Akbarzadeh, M.; Adihou, H.; Hahne, G.; Pobbati, A. V.; Yihui Ng, E.; Guéret, S. M.; Sievers, S.; Pahl, A.; Metz, M. et al.; Zinken, S.; Dötsch, L.; Nowak, C.; Thavam, S.; Friese, A.; Kang, C.; Hong, W.; Waldmann, H.: Discovery of Covalent Inhibitors Targeting the Transcriptional Enhanced Associate Domain Central Pocket. Journal of Medicinal Chemistry 63 (20), pp. 11972 - 11989 (2020)

`T Hart, P.; Hommen, P.; Noisier, A.; Krzyzanowski, A.; Schüler, D.; Porfetye, A. T.; Akbarzadeh, M.; Vetter, I. R.; Adihou, H.; Waldmann, H.: Structure based design of bicyclic peptide inhibitors of RbAp48. Angewandte Chemie International Edition 60 (4), pp. 1813 - 1820 (2020)

`T Hart, P.; Hommen, P.; Noisier, A.; Krzyzanowski, A.; Schüler, D.; Porfetye, A. T.; Akbarzadeh, M.; Vetter, I. R.; Adihou, H.; Waldmann, H.: Structure based design of bicyclic peptide inhibitors of RbAp48. Angewandte Chemie 133 (4), pp. 1841 - 1848 (2020)

Shaaban, S.; Davies, C.; Waldmann, H.: Applications of Chiral Cyclopentadienyl (Cp-x) Metal Complexes in Asymmetric Catalysis. European Journal of Organic Chemistry, pp. 1 - 14 (2020)

Kawamura, T.; Futamura, Y.; Shang, E.; Muroi , M.; Janning, P.; Ueno, M.; Wilke, J.; Takeda, S.; Kondoh , Y.; Ziegler, S. et al.; Watanabe , N.; Waldmann, H.; Osada , H.: Discovery of small-molecule modulator of heterotrimeric G i-protein by integrated phenotypic profiling and chemical proteomics. BioScience, Biotechnology & Biochemistry, pp. 1 - 7 (2020)

Grigalunas, M.; Burhop, A.; Christoforow, A.; Waldmann, H.: Pseudo-natural products and natural product-inspired methods in chemical biology and drug discovery. Current Opinion in Chemical Biology 56, pp. 111 - 118 (2020)

Shaaban, S.; Davies, C.; Merten, C.; Flegel, J.; Otte, F.; Strohmann, C.; Waldmann, H.: Rh(III)-catalyzed C-H Activation of Aryl-Hydroxamates for the Synthesis of Isoindolinones. Chemistry – A European Journal 26 (47), pp. 10729 - 10734 (2020)